Double-Blind Comparison of the Two Hallucinogens Dextromethorphan and Psilocybin: Experience-Dependent and Enduring Psychological Effects in Healthy Volunteers

This double-blind experimental study (n=20) compares the effects of high-dose dextromethorphan (DXM; 400mg/70kg) to psilocybin (10, 20, 30mg/70kg) under conditions typical of therapeutic psychedelic trials. DXM and psilocybin showed increases over placebo in ratings of experiences predictive of psychological benefit at 1 week. However, psilocybin’s effects were dose-dependent and more favourable, while DXM had poorer physical tolerability.

Abstract of Double-Blind Comparison of the Two Hallucinogens Dextromethorphan (DXM) & Psilocybin

Rationale: N-methyl-D-aspartate receptor-mediated dissociatives and serotonergic hallucinogens are being increasingly used in therapeutic interventions that involve nonordinary states of consciousness and may represent a unique mental health paradigm wherein pharmacologically induced experiences are conducive to psychological well-being.

Objective: The aim of this study was to further understand how the phenomenological and health-promoting effects of high-dose dextromethorphan (DXM) compared to psilocybin in the same participants when administered under experimental conditions that are typical of therapeutic psychedelic trials.

Methods: Single, acute oral doses of DXM (400 mg/70 kg), psilocybin (10, 20, 30 mg/70 kg), and inactive placebo were administered under double-blind and psychologically supportive conditions to 20 healthy participants with histories of hallucinogen use. Ratings of personal meaning, spiritual significance, psychological challenge, and psychological insight attributed to acute drug experiences were assessed 7 h (at session end) and 1 week after each drug administration. Persisting psychological effects were assessed 1 week after each drug administration.

Results: High-dose DXM and psilocybin produced similar increases over placebo in ratings of drug experience that was predictive of psychological benefit at 1 week, even when expectancy effects were minimized. These effects tended to favor psilocybin in a dose-dependent manner and were limited by poor physical tolerability for DXM.

Conclusions: This analysis suggests the utility of exploring clinical applications of dissociatives that occur within the supportive contexts that are characteristic of psychedelic research and that prioritize the optimization of psychologically valuable drug experiences.”

Authors: David S. Mathai, Samantha Hilbert, Nathan D. Sepeda, Justin C. Strickland, Roland R. Griffiths & Albert Garcia-Romeu

Summary of Double-Blind Comparison of the Two Hallucinogens Dextromethorphan (DXM) & Psilocybin

Classic serotonergic hallucinogens and N-methyl-D-aspartate receptor-mediated dissociative hallucinogens are being explored as groundbreaking treatments for depression and other psychiatric conditions. These drugs may share downstream mechanisms of action that involve changes in cortical network activity and glutamate-driven neuroplasticity.

Efforts have been made to clarify the psychological effects of classic psychedelics, such as mystical-type experiences, but not all participants who achieve clinical benefit have these canonical experiences. It is, therefore, necessary to categorize drug experiences in ways that are less circumscribed but nonetheless indicative of personal value.

This report presents new data and mixed-methods analyses from a previously conducted double-blind, within-subjects crossover study where hallucinogen-experienced volunteers received doses of oral placebo, DXM, and psilocybin. DXM produced greater disembodiment and physical discomfort than psilocybin.

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Double-Blind Comparison of the Two Hallucinogens Dextromethorphan and Psilocybin: Experience-Dependent and Enduring Psychological Effects in Healthy Volunteers

https://doi.org/10.1089/psymed.2023.0035

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Cite this paper (APA)

Mathai, D. S., Hilbert, S., Sepeda, N. D., Strickland, J. C., Griffiths, R. R., & Garcia-Romeu, A. (2023). Double-Blind Comparison of the Two Hallucinogens Dextromethorphan and Psilocybin: Experience-Dependent and Enduring Psychological Effects in Healthy Volunteers. Psychedelic Medicine.

Study details

Compounds studied
Psilocybin

Topics studied
Healthy Subjects

Study characteristics
Original Re-analysis Active Placebo Double-Blind Within-Subject Randomized

Participants
20 Humans

Authors

Authors associated with this publication with profiles on Blossom

Roland Griffiths
Roland R. Griffiths is one of the strongest voices in psychedelics research. With over 400 journal articles under his belt and as one of the first researchers in the psychedelics renaissance, he has been a vital part of the research community.

Institutes

Institutes associated with this publication

Johns Hopkins University
Johns Hopkins University (Medicine) is host to the Center for Psychedelic and Consciousness Research, which is one of the leading research institutes into psychedelics. The center is led by Roland Griffiths and Matthew Johnson.

Compound Details

The psychedelics given at which dose and how many times

Psilocybin 10 - 30
mg | 3x

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